Publications of Steffen Gaali

Buffa, V.; Meyners, C.; Sugiarto, W. O.; Bauder, M.; Gaali, S.; Hausch, F.: 1,4-Pyrazolyl-Containing SAFit-Analogues are Selective FKBP51 Inhibitors With Improved Ligand Efficiency and Drug-Like Profile. CHEMMEDCHEM (2024)

Gaali, S.; Feng, X.; Hähle, A.; Sippel, C.; Bracher, A.; Hausch, F.: Rapid, Structure-Based Exploration of Pipecolic Acid Amides as Novel Selective Antagonists of the FK506-Binding Protein 51. JOURNAL OF MEDICINAL CHEMISTRY 59 (6), pp. 2410 - 2422 (2016)

Gaali, S.; Kirschner, A.; Cuboni, S.; Hartmann, J.; Kozany, C.; Balsevich, G.; Namendorf, C.; Fernandez-Vizarra, P.; Sippel, C.; Zannas, A. S. et al.; Draenert, R.; Binder, E. B.; Almeida, O. F. X.; Ruehter, G.; Uhr, M.; Schmidt, M. V.; Touma, C.; Bracher, A.; Hausch, F.: Selective inhibitors of the FK506-binding protein 51 by induced fit. NATURE CHEMICAL BIOLOGY 11 (1), pp. 33 - + (2015)

Hartmann, J.; Wagner, K. V.; Gaali, S.; Kirschner, A.; Kozany, C.; Ruhter, G.; Dedic, N.; Häusl, A. S.; Hoeijmakers, L.; Westerholz, S. et al.; Namendorf, C.; Gerlach, T.; Uhr, M.; Chen, A.; Deussing, J. M.; Holsboer, F.; Hausch, F.; Schmidt, M. V.: Pharmacological Inhibition of the Psychiatric Risk Factor FKBP51 Has Anxiolytic Properties. The Journal of neuroscience: the official journal of the Society for Neuroscience 35 (24), pp. 9007 - 16 (2015)

Gaali, S.; Gopalakrishnan, R.; Wang, Y.; Kozany, C.; Hausch, F.: The Chemical Biology of Immunophilin Ligands. Current Medicinal Chemistry 18 (35), pp. 5355 - 5379 (2011)

Gaali, S.; Kozany, C.; Hoogeland, B.; Klein, M.; Hausch, F.: Development of fluorescence polarisation assays for the immunophilins FKBP51/52 and Cyp40. Pharmacopsychiatry 44 (6), p. 290 - 290 (2011)

Gaali, S.; Kozany, C.; Hoogeland, B.; Klein, M.; Hausch, F.: Facile Synthesis of a Fluorescent Cyclosporin A Analogue To Study Cyclophilin 40 and Cyclophilin 18 Ligands. ACS Medicinal Chemistry Letters 1 (9), pp. 536 - 539 (2010)

Gaali, S. P.-G.: Design and synthesis of selective ligands for the FK506-binding protein 51. Dissertation, Ludwig-Maximilians-Universität München, München (2012)